1
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Sokolova A.S.
, Yarovaya O.I.
, Artyushin O.I.
, Sharova E.V.
, Baev D.S.
, Mordvinova E.D.
, Shcherbakov D.N.
, Shnaider T.A.
, Nikitina T.V.
, Esaulkova I.L.
, Ilyina P.A.
, Zarubaev V.V.
, Brel V.K.
, Tolstikova T.G.
, Salakhutdinov N.F.
Design, Synthesis and Antiviral Evaluation of Novel Conjugates of the 1,7,7‐trimethylbicyclo[2.2.1]heptane Scaffold and Saturated N‐heterocycles via 1,2,3‐triazole Linker
Archiv der Pharmazie. 2024.
V.357. N3. e2300549
:1-14. DOI: 10.1002/ardp.202300549
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2
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Yarovaya O.I.
, Filimonov A.S.
, Baev D.S.
, Borisevich S.S.
, Zaykovskaya A.V.
, Chirkova V.Y.
, Marenina M.K.
, Meshkova Y.V.
, Belenkaya S.V.
, Shcherbakov D.N.
, Gureev M.A.
, Luzina O.A.
, Pyankov O.V.
, Salakhutdinov N.F.
, Khvostov M.V.
The Potential of Usnic-Acid-Based Thiazolo-Thiophenes as Inhibitors of the Main Protease of SARS-CoV-2 Viruses
Viruses. 2024.
V.16. N2. 215
:1-20. DOI: 10.3390/v16020215
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3
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Sokolova A.S.
, Baev D.S.
, Mordvinova E.D.
, Yarovaya O.I.
, Volkova N.V.
, Shcherbakov D.N.
, Okhina A.A.
, Rogachev A.D.
, Shnaider T.A.
, Chvileva A.S.
, Nikitina T.V.
, Tolstikova T.G.
, Salakhutdinov N.F.
(+)-fenchol and (-)-isopinocampheol derivatives targeting the entry process of filoviruses
European Journal of Medicinal Chemistry. 2024.
V.275. 116596
. DOI: 10.1016/j.ejmech.2024.116596
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4
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Cheremnych K.P.
, Baev D.S.
, Nacharova E.A.
, Pokrovskii M.A.
, Savelyev V.A.
, Meshkova Y.V.
, Marenina M.K.
, Tolstikova T.G.
, Pokrovski A.G.
, Shults E.E.
Aminocarbonylation of 2-(N-substituted) 5-iodobenzoates: synthesis of glyoxylamido-anthranilates, their cytotoxicity and molecular modeling study
Chemical Papers. 2024.
V.78. N9. P.5639-5656. DOI: 10.1007/s11696-024-03508-0
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5
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Yarovaya O.I.
, Baev D.S.
, Kovaleva K.S.
, Gatilov Y.V.
, Meshkova Y.V.
, Marinina M.K.
, Oreshko V.V.
, Tolstikova T.G.
, Salakhutdinov N.F.
Synthesis and Properties of New Conjugates of Isatin and Bicyclic Monoterpenes
Russian Journal of General Chemistry. 2024.
V.94. N1. P.81-92. DOI: 10.1134/S1070363224010080
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6
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Yarovaya O.I.
, Filimonov A.S.
, Baev D.S.
, Borisevich S.S.
, Chirkova V.Y.
, Zaykovskaya A.V.
, Mordvinova E.D.
, Belenkaya S.V.
, Shcherbakov D.N.
, Luzina O.A.
, Pyankov O.V.
, Salakhutdinov N.F.
Usnic Acid Based Thiazole-Hydrazones as Multi-Targeting Inhibitors of a Wide Spectrum of SARS-CoV-2 Viruses
New Journal of Chemistry. 2023.
V.47. N43. P.19865-19879. DOI: 10.1039/d3nj03598k
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7
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Соколова А.С.
, Баранова Д.В.
, Яровая О.И.
, Зыбкина А.В.
, Мордвинова Е.Д.
, Зайковская А.В.
, Баев Д.С.
, Толстикова Т.Г.
, Щербаков Д.Н.
, Пьянков О.В.
, Максютов Р.А.
, Салахутдинов Н.Ф.
Синтез (1S)-(+)-камфора-10-сульфонамидов и исследование их антифиловирусной активности
Известия Академии наук. Серия химическая. 2023.
Т.72. №10. С.2536-2547. DOI: 10.1007/s11172-023-4056-y
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8
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Cheremnykh K.P.
, Bryzgalov A.O.
, Baev D.S.
, Borisov S.A.
, Sotnikova Y.S.
, Savelyev V.A.
, Tolstikova T.G.
, Sagdullaev S.S.
, Shults E.E.
Synthesis, Pharmacological Evaluation, and Molecular Modeling of Lappaconitine–1,5-Benzodiazepine Hybrids
Molecules. 2023.
V.28. N10. 4234
. DOI: 10.3390/molecules28104234
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9
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Далингер А.И.
, Баев Д.С.
, Яровая О.И.
, Чиркова В.Ю.
, Шарлаева Е.А.
, Беленькая С.В.
, Щербаков Д.Н.
, Салахутдинов Н.Ф.
, Вацадзе С.З.
Синтез несимметричных амидов N-бензилбиспидинола и изучение их ингибирующей активности по отношению к основной вирусной протеазе SARS-CoV-2
Известия Академии наук. Серия химическая. 2023.
Т.72. №1. С.239-247. DOI: 10.1007/s11172-023-3729-x
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10
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Baev D.S.
, Blokhin M.E.
, Chirkova V.Y.
, Belenkaya S.V.
, Luzina O.A.
, Yarovaya O.I.
, Salakhutdinov N.F.
, Shcherbakov D.N.
Triterpenic Acid Amides as Potential Inhibitors of the SARS-CoV-2 Main Protease
Molecules. 2023.
V.28. N1. 303
. DOI: 10.3390/molecules28010303
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11
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Filimonov A.S.
, Yarovaya O.I.
, Zaykovskaya A.V.
, Rudometova N.B.
, Shcherbakov D.N.
, Chirkova V.Y.
, Baev D.S.
, Borisevich S.S.
, Luzina O.A.
, Pyankov O.V.
, Maksyutov R.A.
, Salakhutdinov N.F.
(+)-Usnic Acid and Its Derivatives as Inhibitors of a Wide Spectrum of SARS-CoV-2 Viruses
Viruses. 2022.
V.14. N10. 2154
. DOI: 10.3390/v14102154
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12
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Shcherbakov D.
, Baev D.
, Kalinin M.
, Dalinger A.
, Chirkova V.
, Belenkaya S.
, Khvostov A.
, Krut'ko D.
, Medved'ko A.
, Volosnikova E.
, Sharlaeva E.
, Shanshin D.
, Tolstikova T.
, Maksyutov R.
, Yarovaya O.
, Salakhutdinov N.
, Vatsadze S.
Design and Evaluation of Bispidine-Based SARS-CoV-2 Main Protease Inhibitors
ACS Medicinal Chemistry Letters. 2022.
V.13. N1. P.140-147. DOI: 10.1021/acsmedchemlett.1c00299
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13
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Reshetnikov D.V.
, Ivanov I.D.
, Baev D.S.
, Rybalova T.V.
, Mozhaitsev E.S.
, Patrushev S.S.
, Vavilin V.A.
, Tolstikova T.G.
, Shults E.E.
Design, Synthesis and Assay of Novel Methylxanthine–Alkynylmethylamine Derivatives as Acetylcholinesterase Inhibitors
Molecules. 2022.
V.27. N24. 8787
. DOI: 10.3390/molecules27248787
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